THE UNITS OF CHEMICAL AND PHARMACEUTICAL SCIENCE (DSCF) AND LIFE SCIENCES (DSV) HAVE DIFFERENTIATED AND COMPLEMENTARY SKILLS AND ROLES. UNITS-DSCF CURRENT THE DESIGN, SYNTHESIS AND MODIFICATION OF NEW DEUBILIQUITINASI (ISISIDASEI) INHIBITORS WHICH ARE STRUCTURALLY RELATED TO THIS 2CPE INHIBITOR, THE ACTIVITY OF WHICH HAS BEEN RECENTLY DEMONSTRATED IN VITRO AND IN VIVO. THE DESIGN OF SECOND GENERATION INHIBITORS WILL INFORM THE